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Contraindicated. Cobicistat can be a CYP3A4 inhibitor; contraindicated with CYP3A4 substrates for which elevated plasma concentrations are linked to major and/or lifestyle-threatening occasions.Keep an eye on Carefully (1)crofelemer raises amounts of ergotamine by impacting hepatic/intestinal enzyme CYP3A4 metabolism. Use Caution/Watch. Crofelemer